31. Thermosensitive transient receptor potential channels in human corneal epithelial cells
    2010/11/10 by Stefan Mergler, Fabian Garreis, Monika Sahlmüller +3 · 25 citations
    Biochemistry, Genetics and Molecular Biology · Chemistry · Neuroscience · #Agonist #Biochemistry #Biology #Biophysics #Calcium #Capsazepine #Cell biology #Channel blocker #Chemistry #Connexins and lens biology #Intracellular #Ion Channels and Receptors #Ionomycin #Membrane potential #Neurobiology and Insect Physiology Research #Patch clamp #Receptor #Ruthenium red #TRPC #TRPC6 #TRPM8 #TRPV #TRPV1 #TRPV4 #Transient receptor potential channel
32. ApoE Promotes the Proteolytic Degradation of Aβ
    2008/06/01 by Qingguang Jiang, C.Y. Daniel Lee, Shweta Mandrekar +18 · 2 citations
    Chemistry · Medicine · Neuroscience · #Agonist #Alzheimer's disease research and treatments #Apolipoprotein E #Autophagy #Biochemistry #Biology #Cell biology #Chemistry #Cholesterol and Lipid Metabolism #Disease #Drug Transport and Resistance Mechanisms #Endocrinology #Enzyme #Inflammation #Insulin-degrading enzyme #Internal medicine #Lipid-anchored protein #Medicine #Microglia #Neprilysin #Neuroinflammation #Neuroscience #Receptor
33. Non-redundant Functions of Cyclooxygenases: Oxygenation of Endocannabinoids
    2008/02/05 by Carol A. Rouzer, Lawrence J. Marnett · 1 citation
    Biochemistry, Genetics and Molecular Biology · Chemistry · Medicine · #Agonist #Arachidonic acid #Biochemistry #Biosynthesis #Cannabis and Cannabinoid Research #Chemistry #Cyclooxygenase #Eicosanoids and Hypertension Pharmacology #Endocannabinoid system #Enzyme #Inflammatory mediators and NSAID effects #Internal medicine #Lipid signaling #Medicine #Platelet #Prostaglandin #Receptor #Thromboxane #Thromboxane A2
34. Denufosol: A review of studies with inhaled P2Y2 agonists that led to Phase 3
    2008/01/02 by Donald Kellerman, Donald J. Kellerman, Andrea Rossi Mospan +6 · 1 citation
    Medicine · #Adverse effect #Agonist #Anesthesia #Cystic Fibrosis Research Advances #Cystic fibrosis #Inhalation and Respiratory Drug Delivery #Internal medicine #Lung #Medicine #Mucociliary clearance #Nebulizer #Pathology #Pharmacokinetics #Pharmacology #Placebo #Receptor #Respiratory system #Tracheal and airway disorders
35. The diverse CB1and CB2receptor pharmacology of three plant cannabinoids: Δ9‐tetrahydrocannabinol, cannabidiol and Δ9‐tetrahydrocannabivarin
    2007/09/10 by R G Pertwee, Roger G. Pertwee · 54 citations
    Agricultural and Biological Sciences · Chemistry · Medicine · Neuroscience · #Agonist #Biochemistry #Biology #Cannabidiol #Cannabinoid #Cannabinoid Receptor Agonists #Cannabinoid receptor #Cannabinoid receptor antagonist #Cannabinoid receptor type 2 #Cannabis #Cannabis and Cannabinoid Research #Chemistry #Competitive antagonist #GABA and Rice Research #Medicine #Partial agonist #Pharmacology #Receptor #Sleep and Wakefulness Research
36. The MC4 receptor and control of appetite
    2006/10/17 by Roger A.H. Adan, R A H Adan, B Tiesjema +9 · 26 citations
    Biochemistry, Genetics and Molecular Biology · Medicine · Neuroscience · Nursing · #Agonist #Anorectic #Appetite #Biochemical Analysis and Sensing Techniques #Biology #Endocrinology #Food intake #Hypothalamus #Internal medicine #Meal #Medicine #Melanocortin #Melanocortin 4 receptor #Obesity #Pharmacology #Receptor #Regulation of Appetite and Obesity #melanin and skin pigmentation
37. Association of Dopamine Agonist Use With Impulse Control Disorders in Parkinson Disease
    2006/07/01 by Daniel Weintraub, Andrew D. Siderowf, Andrew Siderowf +7 · 32 citations
    Medicine · Psychology · #Agonist #Disease #Dopamine #Dopamine agonist #Dopaminergic #Hypersexuality #Impulse control disorder #Internal medicine #Medicine #Neurological disorders and treatments #Parkinson's Disease Mechanisms and Treatments #Parkinson's disease #Pathological #Psychiatry #Psychology #Restless Legs Syndrome Research #Ropinirole
38. Levels of apoptosis in human granulosa cells seem to be comparable after therapy with a gonadotropin-releasing hormone agonist or antagonist
    2006/02/01 by Franca Giampietro, Silvia Sancilio, Gian Mario Tiboni +2 · 8 citations
    Chemistry · Immunology and Microbiology · Medicine · #Agonist #Antagonist #Apoptosis #Buserelin #Chemistry #Endocrinology #Gonadotropin #Gonadotropin-releasing hormone #Gonadotropin-releasing hormone agonist #Gonadotropin-releasing hormone antagonist #Hormone #Hormone antagonist #Internal medicine #Luteinizing hormone #Medicine #Ovarian function and disorders #Receptor #Reproductive Biology and Fertility #Reproductive System and Pregnancy
39. Distinct rhythm generators for inspiration and expiration in the juvenile rat
    2005/11/17 by Wiktor A. Janczewski, Jack L. Feldman · 3 citations
    Neuroscience · Psychology · Medicine · #Neuroscience of respiration and sleep #Neuroendocrine regulation and behavior #Sleep and Wakefulness Research #Rhythm #Expiration #Brainstem #Reflex #Neuroscience #Agonist #Respiratory system #Medicine #Anatomy #Anesthesia #Biology #Internal medicine #Receptor
40. Trace amines reduce GABAB receptor-mediated presynaptic inhibition at GABAergic synapses of the rat substantia nigra pars compacta
    2005/11/01 by Nicola Berretta, Michela Giustizieri, Giorgio Bernardi +2 · 5 citations
    Biochemistry, Genetics and Molecular Biology · Chemistry · Neuroscience · #Agonist #Amphetamine #Baclofen #Biochemistry #Biology #Chemistry #Dopamine #Dopaminergic #GABAA receptor #GABAB receptor #GABAergic #Inhibitory postsynaptic potential #Neuroscience #Neuroscience and Neuropharmacology Research #Neurotransmitter Receptor Influence on Behavior #Pars compacta #Pharmacology #Receptor #Receptor Mechanisms and Signaling #Substantia nigra
41. Spinal nerve ligation increases α2-adrenergic receptor G-protein coupling in the spinal cord
    2005/02/17 by Carsten Bantel, James C. Eisenach, Frédéric Duflo +3 · 23 citations
    Biochemistry, Genetics and Molecular Biology · Chemistry · Medicine · Neuroscience · #Adrenergic #Adrenergic receptor #Agonist #Antagonist #Biology #Chemistry #Clonidine #Endocrinology #Internal medicine #Ion channel regulation and function #Medicine #Musculoskeletal pain and rehabilitation #Neuropathic pain #Neuroscience #Nociception #Pain Mechanisms and Treatments #Pharmacology #Prazosin #Rauwolscine #Receptor #Spinal cord
42. Ghrelin Stimulates, Whereas Des-Octanoyl Ghrelin Inhibits, Glucose Output by Primary Hepatocytes
    2005/02/01 by Carlotta Gauna, Patric J. D. Delhanty, Leo J. Hofland +7 · 28 citations
    Chemistry · Medicine · Neuroscience · #Adipose Tissue and Metabolism #Agonist #Biochemistry #Biology #Chemistry #Endocrinology #Ghrelin #Growth hormone secretagogue receptor #Hepatocyte #In vitro #Incubation #Insulin #Internal medicine #Medicine #Pancreatic function and diabetes #Receptor #Regulation of Appetite and Obesity #Secretagogue
43. Modulating the Rate and Rhythmicity of Perceptual Rivalry Alternations with the Mixed 5-HT2A and 5-HT1A Agonist Psilocybin
    2005/01/26 by Olivia Carter, Olivia L Carter, John D Pettigrew +9 · 1 citation
    Biochemistry, Genetics and Molecular Biology · Medicine · Neuroscience · Psychology · #Agonist #Cognitive psychology #Hallucinogen #Internal medicine #Medicine #Neuroscience #Neurotransmitter Receptor Influence on Behavior #Nicotinic Acetylcholine Receptors Study #Perception #Psilocybin #Psychedelics and Drug Studies #Psychiatry #Psychology #Receptor #Rivalry
44. Molecular Determinants Involved in the Allosteric Control of Agonist Affinity in the GABAB Receptor by the GABAB2 Subunit
    2004/04/01 by Jianfeng Liu, Damien Maurel, Sébastien Etzol +5 · 2 citations
    Biochemistry, Genetics and Molecular Biology · Chemistry · Neuroscience · Nursing · #Agonist #Allosteric modulator #Allosteric regulation #Biochemical Analysis and Sensing Techniques #Biochemistry #Biology #Biophysics #Chemistry #G alpha subunit #GABAB receptor #Gamma-aminobutyric acid receptor subunit alpha-1 #Gene #Neuroscience #Neuroscience and Neuropharmacology Research #Protein subunit #Receptor #Receptor Mechanisms and Signaling #q-bio.BM #q-bio.NC
45. Adenosine A 3 Receptor Activation Modulates the Capillary Endothelial Glycocalyx
    2003/11/25 by Steven H. Platts, Brian R. Duling · 9 citations
    Biochemistry, Genetics and Molecular Biology · Chemistry · Medicine · #Adenosine #Adenosine receptor #Agonist #Biochemistry #Biology #Blood transfusion and management #Cell biology #Chemistry #Endocrinology #Endothelial stem cell #Endothelium #Glycocalyx #Hemoglobin structure and function #In vitro #Internal medicine #Medicine #Receptor #Trauma, Hemostasis, Coagulopathy, Resuscitation #Vascular permeability
46. Histamine induces cytoskeletal changes in human eosinophils via the H4 receptor
    2003/11/01 by Karen F Buckland, Karen Buckland, Timothy J. Williams +3 · 27 citations
    Chemistry · Immunology and Microbiology · Medicine · #Agonist #Allergic Rhinitis and Sensitization #Antagonist #Asthma and respiratory diseases #Biochemistry #Biology #Chemistry #Endocrinology #Histamine #Histamine H1 receptor #Histamine H2 receptor #Histamine H3 receptor #Histamine H4 receptor #Histamine N-methyltransferase #Histamine receptor #Internal medicine #Mast cells and histamine #Medicine #Pharmacology #Receptor #Thioperamide
47. Endogenous Melanocortin Antagonist in Fish: Structure, Brain Mapping, and Regulation by Fasting of the Goldfish Agouti-Related Protein Gene
    2003/07/08 by José Miguel Cerdá-Reverter, José Miguel Cerdá‐Reverter, Richard Peter +1 · 28 citations
    Medicine · Neuroscience · Nursing · #Adipokines, Inflammation, and Metabolic Diseases #Agonist #Antagonist #Arcuate nucleus #Biochemical Analysis and Sensing Techniques #Biology #Cell biology #Endocrinology #Endogeny #Gene #Gene expression #Genetics #Hormone #Hypothalamus #In situ hybridization #Internal medicine #Medicine #Melanocortin #Melanocortin 3 receptor #Melanocortin 4 receptor #Melanocortin receptor #Neuropeptide #Nucleus #Receptor #Regulation of Appetite and Obesity
48. The Orphan G Protein-coupled Receptors GPR41 and GPR43 Are Activated by Propionate and Other Short Chain Carboxylic Acids
    2003/03/01 by Andrew J. Brown, Susan M. Goldsworthy, Ashley Barnes +26 · 64 citations
    Biochemistry, Genetics and Molecular Biology · Chemistry · Immunology and Microbiology · Neuroscience · #Agonist #Biochemistry #Biology #Chemistry #G protein #G protein-coupled inwardly-rectifying potassium channel #Gene #Immune Cell Function and Interaction #Molecular biology #Neuropeptides and Animal Physiology #Receptor #Receptor Mechanisms and Signaling #Xenopus
49. The open field as a paradigm to measure the effects of drugs on anxiety-like behaviors: a review
    2003/02/01 by Laetitia Prut, L. Prut, Catherine Belzung · 57 citations
    Agricultural and Biological Sciences · Medicine · Neuroscience · Psychology · #Agonist #Alprazolam #Anti-Anxiety Agents #Anxiety #Anxiety disorder #Anxiogenic #Anxiolytic #Benzodiazepine #Generalized anxiety disorder #Internal medicine #Inverse agonist #Medicine #Neuroendocrine regulation and behavior #Neurotransmitter Receptor Influence on Behavior #Open field #Panic disorder #Partial agonist #Pharmacological Effects and Assays #Pharmacology #Psychiatry #Psychology #Receptor
50. The Unique Ligand-binding Pocket for the Human Prostacyclin Receptor
    2003/02/01 by Jeremiah Stitham, Aleksandar Stojanovic, Aleksandar Stojanović +4 · 8 citations
    Biochemistry, Genetics and Molecular Biology · Chemistry · Neuroscience · #Agonist #Amino acid #Biochemistry #Chemistry #Eicosanoids and Hypertension Pharmacology #G protein-coupled receptor #Ligand (biochemistry) #Neuropeptides and Animal Physiology #Prostacyclin #Receptor #Receptor Mechanisms and Signaling #Rhodopsin #Stereochemistry #Transmembrane domain
51. G Protein-coupled Receptor Kinase 5 Regulates β1-Adrenergic Receptor Association with PSD-95
    2002/01/01 by Liaoyuan A. Hu, Wei Chen, Richard T. Premont +2 · 1 citation
    Biochemistry, Genetics and Molecular Biology · Neuroscience · #Agonist #Beta adrenergic receptor kinase #Biochemistry #Biology #Cell biology #G protein-coupled receptor #G protein-coupled receptor kinase #Gene #Immunoprecipitation #Kinase #Mutant #Neuropeptides and Animal Physiology #Neuroscience and Neuropharmacology Research #PDZ domain #Phosphorylation #Protein kinase domain #Receptor #Receptor Mechanisms and Signaling #Signal transduction
52. Force-feeding procedure and physiological indicators of stress in male mule ducks
    2001/12/01 by Daniel D. Guemene, G. Guy, Jérôme Noirault +3 · 3 citations
    Agricultural and Biological Sciences · Medicine · Neuroscience · Veterinary · #Adrenocorticotropic hormone #Agonist #Animal Behavior and Welfare Studies #Animal Nutrition and Physiology #Animal science #Biology #Chronic stress #Corticosterone #Endocrinology #Hormone #Internal medicine #Medicine #Neuroscience #Period (music) #Physics #Receptor #Stress Responses and Cortisol #Stressor
53. NMDA and glycine regulate the affinity of the Mg2+-block site in NR1-1a/NR2A NMDA receptor channels expressed in Xenopus oocytes
    2001/03/01 by Y. Liu, R.H. Hill, Russell H. Hill +4 · 1 citation
    Biochemistry, Genetics and Molecular Biology · Chemistry · Neuroscience · #Agonist #Amino acid #Biochemistry #Biology #Biophysics #Chemistry #Coordination Chemistry and Organometallics #Glutamate receptor #Glycine #Glycine receptor #Ion channel #Ion channel regulation and function #NMDA receptor #Neuroscience and Neuropharmacology Research #Receptor #Xenopus
54. Resveratrol Acts as a Mixed Agonist/Antagonist for Estrogen Receptors α and β*
    2000/10/01 by Jennifer L. Bowers, Valentyn V. Tyulmenkov, Sarah C. Jernigan +2 · 28 citations
    Biochemistry, Genetics and Molecular Biology · Chemistry · Medicine · #Agonist #Antagonist #Biochemistry #Biology #Cancer #Chemistry #Endocrinology #Estrogen #Estrogen and related hormone effects #Estrogen receptor #Estrogen receptor alpha #Estrogen receptor beta #Genomics, phytochemicals, and oxidative stress #Internal medicine #Medicine #Partial agonist #Pharmacology #Phytoestrogens #Receptor #Resveratrol #Sirtuins and Resveratrol in Medicine
55. d -Serine is an endogenous ligand for the glycine site of the N -methyl- d -aspartate receptor
    2000/04/25 by Jean‐Pierre Mothet, Angèle Parent, Herman Wolosker +5 · 2 citations
    Biochemistry, Genetics and Molecular Biology · Neuroscience · Chemistry · #Amino Acid Enzymes and Metabolism #Neuroscience and Neuropharmacology Research #Molecular Sensors and Ion Detection #NMDA receptor #Glycine #Serine #Receptor #Biochemistry #Glutamate receptor #Agonist #Endogeny #Biology #Chemistry #Amino acid #Enzyme
56. Heterodimerization is required for the formation of a functional GABAB receptor
    1998/12/01 by Julia H. White, Alan Wise, Martin J. Main +10 · 8 citations
    Biochemistry, Genetics and Molecular Biology · Chemistry · Immunology and Microbiology · Neuroscience · #5-HT5A receptor #Agonist #Amino acid #Antimicrobial Peptides and Activities #Biochemistry #Biology #Cell biology #Chemistry #Class C GPCR #Enzyme-linked receptor #GABAA receptor #GABAA-rho receptor #GABAB receptor #GABBR1 #Glycine #Glycine receptor #HEK 293 cells #Inhibitory postsynaptic potential #Metabotropic receptor #Neuroscience #Neuroscience and Neuropharmacology Research #Neurotransmitter receptor #Protease-activated receptor 2 #Receptor #Receptor Mechanisms and Signaling
57. Gabaergic Control of Spinal Locomotor Networks in the Neonatal Rat
    1998/11/01 by Jean‐René Cazalets, Sandrine S. Bertrand, Youssef Sqalli-Houssaini +1 · 2 citations
    Neuroscience · Biochemistry, Genetics and Molecular Biology · Psychology · Chemistry · Medicine · #Neuroscience and Neuropharmacology Research #Zebrafish Biomedical Research Applications #Neuroendocrine regulation and behavior #GABAergic #Spinal cord #Muscimol #Locomotor activity #Neuroscience #Lumbar #Lumbar Spinal Cord #GABAA receptor #Baclofen #Chemistry #Biology #Inhibitory postsynaptic potential #Receptor #Agonist #Anatomy #Medicine #Pharmacology #Internal medicine
58. Characterization of the relaxant action of urocortin, a new peptide related to corticotropin‐releasing factor in the rat isolated basilar artery
    1998/11/01 by L Schilling, Lothar Schilling, Ch Kanzler +4 · 6 citations
    Chemistry · Medicine · Neuroscience · Psychology · #Agonist #Apamin #Biochemical effects in animals #Chemistry #Endocrinology #Internal medicine #Medicine #Neuroendocrine regulation and behavior #Potassium channel #Receptor #Stress Responses and Cortisol #Urocortin
59. The neuroactive steroid allopregnanolone suppresses hypothalamic gonadotropin-releasing hormone release through a mechanism mediated by the gamma-aminobutyric acidA receptor
    1998/07/01 by Aldo E. Calogero, AE Calogero, Marco Palumbo +13 · 15 citations
    Chemistry · Medicine · Neuroscience · Psychology · #Agonist #Allopregnanolone #Bicuculline #Biology #Chemistry #Endocrinology #GABAA receptor #Hypothalamic control of reproductive hormones #Internal medicine #Medicine #Neuroactive steroid #Neuroendocrine regulation and behavior #Pregnane #Pregnanolone #Pregnenolone sulfate #Receptor #Stress Responses and Cortisol
60. Human Estrogen Receptor β Binds DNA in a Manner Similar to and Dimerizes with Estrogen Receptor α
    1997/10/01 by Paul Pace, Jacqueline Taylor, Sumathy Suntharalingam +2 · 5 citations
    Biochemistry, Genetics and Molecular Biology · Chemistry · Pharmacology, Toxicology and Pharmaceutics · #Agonist #Bioactive Compounds and Antitumor Agents #Biochemistry #Biology #Chemistry #DNA #DNA and Nucleic Acid Chemistry #Endocrinology #Estrogen #Estrogen and related hormone effects #Estrogen receptor #Estrogen receptor alpha #Estrogen receptor beta #Genetics #Hormone response element #In vitro #Ligand (biochemistry) #Molecular biology #Receptor #Tamoxifen

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