- Pharmacological Profile of Lurasidone, a Novel Antipsychotic Agent with Potent 5-Hydroxytryptamine 7 (5-HT7) and 5-HT1A Receptor Activity
2010/04/20 by Tadashi Ishibashi, Tomoko Horisawa, Kumiko Tokuda +15 · 29 citations
Biochemistry, Genetics and Molecular Biology · Chemistry · Medicine · Neuroscience · #5-HT receptor #Agonist #Antipsychotic #Atypical antipsychotic #Biochemistry #Biology #Chemistry #Dopamine receptor D2 #Lurasidone #Medicine #Neuroscience and Neuropharmacology Research #Neurotransmitter Receptor Influence on Behavior #Partial agonist #Pharmacological Receptor Mechanisms and Effects #Pharmacology #Receptor #Serotonin
- The diverse CB1and CB2receptor pharmacology of three plant cannabinoids: Δ9‐tetrahydrocannabinol, cannabidiol and Δ9‐tetrahydrocannabivarin
2007/09/10 by Roger G. Pertwee, R G Pertwee · 54 citations
Agricultural and Biological Sciences · Chemistry · Medicine · Neuroscience · #Agonist #Biochemistry #Biology #Cannabidiol #Cannabinoid #Cannabinoid Receptor Agonists #Cannabinoid receptor #Cannabinoid receptor antagonist #Cannabinoid receptor type 2 #Cannabis #Cannabis and Cannabinoid Research #Chemistry #Competitive antagonist #GABA and Rice Research #Medicine #Partial agonist #Pharmacology #Receptor #Sleep and Wakefulness Research
- Functional Selectivity and Classical Concepts of Quantitative Pharmacology
2006/06/28 by Jonathan D. Urban, William P. Clarke, Mark von Zastrow +11 · 45 citations
Biochemistry, Genetics and Molecular Biology · Chemistry · Neuroscience · Pharmacology, Toxicology and Pharmaceutics · #Agonist #Biochemistry #Biology #Cell biology #Chemistry #Computational biology #Functional selectivity #G protein-coupled receptor #Intrinsic activity #Mechanism (biology) #Molecular Pharmacology #Neuropeptides and Animal Physiology #Neuroscience #Partial agonist #Pharmacogenetics and Drug Metabolism #Pharmacology #Receptor #Receptor Mechanisms and Signaling #Signal transduction
- The open field as a paradigm to measure the effects of drugs on anxiety-like behaviors: a review
2003/02/01 by Laetitia Prut, L. Prut, Catherine Belzung · 57 citations
Agricultural and Biological Sciences · Medicine · Neuroscience · Psychology · #Agonist #Alprazolam #Anti-Anxiety Agents #Anxiety #Anxiety disorder #Anxiogenic #Anxiolytic #Benzodiazepine #Generalized anxiety disorder #Internal medicine #Inverse agonist #Medicine #Neuroendocrine regulation and behavior #Neurotransmitter Receptor Influence on Behavior #Open field #Panic disorder #Partial agonist #Pharmacological Effects and Assays #Pharmacology #Psychiatry #Psychology #Receptor
- Resveratrol Acts as a Mixed Agonist/Antagonist for Estrogen Receptors α and β*
2000/10/01 by Jennifer L. Bowers, Valentyn V. Tyulmenkov, Sarah Jernigan +2 · 28 citations
Biochemistry, Genetics and Molecular Biology · Chemistry · Medicine · #Agonist #Antagonist #Biochemistry #Biology #Cancer #Chemistry #Endocrinology #Estrogen #Estrogen and related hormone effects #Estrogen receptor #Estrogen receptor alpha #Estrogen receptor beta #Genomics, phytochemicals, and oxidative stress #Internal medicine #Medicine #Partial agonist #Pharmacology #Phytoestrogens #Receptor #Resveratrol #Sirtuins and Resveratrol in Medicine
- Role of 5‐ht7 receptors in the long‐lasting hypotensive response induced by 5‐hydroxytryptamine in the rat
1997/05/01 by José A. Terrón · 19 citations
Chemistry · Medicine · Neuroscience · Psychology · #5-HT receptor #Agonist #Antagonist #Chemistry #Dopamine agonist #Endocrinology #Internal medicine #Ketanserin #Lisuride #Medicine #Metergoline #Methysergide #Neuroendocrine regulation and behavior #Neuroscience and Neuropharmacology Research #Neurotransmitter Receptor Influence on Behavior #Partial agonist #Pharmacology #Receptor #Ritanserin #Serotonin