International Union of Basic and Clinical Pharmacology. XCVII. G Protein–Coupled Estrogen Receptor and Its Pharmacologic Modulators

2015/05/29 by Eric R. Prossnitz, Jeffrey B. Arterburn · 6 citations
Biochemistry, Genetics and Molecular Biology · Pharmacology, Toxicology and Pharmaceutics · #Estrogen and related hormone effects #Pharmacogenetics and Drug Metabolism #Receptor Mechanisms and Signaling

paper · pdf · doi:10.1124/pr.114.009712

openalex publication_date 2015/05/29 · crossref created 2015/05/29 · crossref issued 2015/07/01 · crossref published 2015/07/01 · crossref published-print 2015/07/01 · crossref deposited 2025/02/18 · openalex created_date 2025/10/10 · openalex updated_date 2026/08/04 · crossref indexed 2026/08/04

Citations

• G Protein-Coupled Receptor 30 Localizes to the Endoplasmic Reticulum and Is Not Activated by Estradiol
• The structure and function of G-protein-coupled receptors
• Development of subtype-selective oestrogen receptor-based therapeutics
• Estrogen receptor β selective nonsteroidal estrogens: seeking clinical indications
• Membrane Estrogen Receptor Regulation of Hypothalamic Function
• Estrogen: A master regulator of bioenergetic systems in the brain and body
• Estrogen Carcinogenesis in Breast Cancer
• Estrogen receptors alpha (ERα) and beta (ERβ): Subtype-selective ligands and clinical potential
• Estrogen Receptors: Therapies Targeted to Receptor Subtypes
• Coregulator Function: A Key to Understanding Tissue Specificity of Selective Receptor Modulators
• Structure-Function of the G Protein–Coupled Receptor Superfamily
• International Union of Pharmacology. LXIV. Estrogen Receptors
• Cloning of a novel receptor expressed in rat prostate and ovary.
• Comparison of the Ligand Binding Specificity and Transcript Tissue Distribution of Estrogen Receptors α and β
• Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction
• The G-protein-coupled estrogen receptor GPER in health and disease
• Estrogen receptor protein content is different in abdominal than gluteal subcutaneous adipose tissue of overweight-to-obese premenopausal women
• Estrogen and the cardiovascular system
• GPR30, but not estrogen receptor-α, is crucial in the treatment of experimental autoimmune encephalomyelitis by oral ethinyl estradiol
• Endocrine Disruptors: From Endocrine to Metabolic Disruption
• Estrogens and health in males
• Quantitative Structure-Activity Relationship of Various Endogenous Estrogen Metabolites for Human Estrogen Receptor α and β Subtypes: Insights into the Structural Determinants Favoring a Differential Subtype Binding

Cited by

• Estrogen Signaling as a Therapeutic Target in Neurodevelopmental Disorders
• Alfatradiol [wikipedia]
• Estriol (medication) [wikipedia]
• Estrone (medication) [wikipedia]
• Ethinylestradiol [wikipedia]
• Pharmacodynamics of estradiol [wikipedia]