Estrogen receptors alpha (ERα) and beta (ERβ): Subtype-selective ligands and clinical potential

2014/06/24 by Ilaria Paterni, Carlotta Granchi, John A. Katzenellenbogen +1 · 2 citations
Biochemistry, Genetics and Molecular Biology · Neuroscience · #Estrogen and related hormone effects #Nuclear Receptors and Signaling #Retinoids in leukemia and cellular processes

paper · doi:10.1016/j.steroids.2014.06.012

openalex publication_date 2014/06/24 · crossref created 2014/06/24 · crossref issued 2014/11/01 · crossref published 2014/11/01 · crossref published-print 2014/11/01 · crossref deposited 2022/04/09 · openalex created_date 2025/10/10 · openalex updated_date 2026/08/01 · crossref indexed 2026/08/05

Citations

• Estrogenic hormone action in the heart: regulatory network and function
• Development of subtype-selective oestrogen receptor-based therapeutics
• PET-based estradiol challenge as a predictive biomarker of response to endocrine therapy in women with estrogen-receptor-positive breast cancer
• Estrogen Receptors: Therapies Targeted to Receptor Subtypes
• International Union of Pharmacology. LXIV. Estrogen Receptors
• Comparison of the Ligand Binding Specificity and Transcript Tissue Distribution of Estrogen Receptors α and β
• Structural Evolutions of Salicylaldoximes as Selective Agonists for Estrogen Receptor β
• Protective actions of sex steroid hormones in Alzheimer’s disease
• The androgen derivative 5α-androstane-3β,17β-diol inhibits tumor necrosis factor α and lipopolysaccharide induced inflammatory response in human endothelial cells and in mice aorta
• Molecular basis of agonism and antagonism in the oestrogen receptor
• Antiestrogens and Selective Estrogen Receptor Modulators as Multifunctional Medicines. 2. Clinical Considerations and New Agents
• Evaluation of an Estrogen Receptor-β Agonist in Animal Models of Human Disease

Cited by

• International Union of Basic and Clinical Pharmacology. XCVII. G Protein–Coupled Estrogen Receptor and Its Pharmacologic Modulators
• Estrogen receptor alpha [wikipedia]