Allosteric Ligands of the Glucagon-Like Peptide 1 Receptor (GLP-1R) Differentially Modulate Endogenous and Exogenous Peptide Responses in a Pathway-Selective Manner: Implications for Drug Screening

2010/06/15 by Cassandra Koole, Denise Wootten, John Simms +8 · 3 citations
Medicine · Biochemistry, Genetics and Molecular Biology · Neuroscience · #Diabetes Treatment and Management #Receptor Mechanisms and Signaling #Neuropeptides and Animal Physiology

paper · doi:10.1124/mol.110.065664

Citations

• Functional Selectivity and Classical Concepts of Quantitative Pharmacology

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