Seven Transmembrane Receptors as Shapeshifting Proteins: The Impact of Allosteric Modulation and Functional Selectivity on New Drug Discovery

2010/05/14 by Terry Kenakin, Laurence J. Miller · 6 citations
Biochemistry, Genetics and Molecular Biology · Neuroscience · #Receptor Mechanisms and Signaling #Neuroscience and Neuropharmacology Research #Chemical Synthesis and Analysis

paper · doi:10.1124/pr.108.000992

Citations

• Evolving Concepts in G Protein-Coupled Receptor Endocytosis: The Role in Receptor Desensitization and Signaling
• Structural Mechanisms for Domain Movements in Proteins

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