Parallel Functional Activity Profiling Reveals Valvulopathogens Are Potent 5-Hydroxytryptamine2B Receptor Agonists: Implications for Drug Safety Assessment

2009/07/02 by Xi‐Ping Huang, Xi-Ping Huang, Vincent Setola +10 · 3 citations
Medicine · #Pharmacology and Obesity Treatment #Atrial Fibrillation Management and Outcomes #Cardiac Arrhythmias and Treatments

paper · doi:10.1124/mol.109.058057

Citations

• Possible Role of Valvular Serotonin 5-HT2B Receptors in the Cardiopathy Associated with Fenfluramine
• Functional Selectivity and Classical Concepts of Quantitative Pharmacology

Cited by

• International Union of Basic and Clinical Pharmacology. CX. Classification of Receptors for 5-hydroxytryptamine; Pharmacology and Function
• Microdosing psychedelics and the risk of cardiac fibrosis and valvulopathy: Comparison to known cardiotoxins
• Molecular design of a therapeutic LSD analogue with reduced hallucinogenic potential