5-Aza-4′-thio-2′-deoxycytidine, a New Orally Bioavailable Nontoxic “Best-in-Class”: DNA Methyltransferase 1–Depleting Agent in Clinical Development

2021/09/09 by William B. Parker, Jaideep V. Thottassery · 16 citations
Biochemistry, Genetics and Molecular Biology · Chemistry · Medicine · #Acute Lymphoblastic Leukemia research #Azacitidine #Biochemistry #Biology #Cancer #Chemistry #DNA #DNA methylation #DNA methyltransferase #DNMT1 #Decitabine #Deoxycytidine #Epigenetics and DNA Methylation #Genetics #Hemoglobinopathies and Related Disorders #Methylation #Methyltransferase #Pharmacology

paper · pdf · doi:10.1124/jpet.121.000758

openalex publication_date 2021/09/09 · openalex created_date 2025/10/10 · openalex updated_date 2026/08/06

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