5α-Reduction of norethisterone enhances its binding affinity for androgen receptors but diminishes its androgenic potency

1997/01/01 by Ana E. Lemus, Juana Enríquez, Gustavo A. García +4 · 1 citation
Biochemistry, Genetics and Molecular Biology · Medicine · #Estrogen and related hormone effects #Hormonal and reproductive studies #Prostate Cancer Treatment and Research

paper · doi:10.1016/s0960-0760(96)00172-0

crossref issued 1997/01/01 · crossref published 1997/01/01 · crossref published-print 1997/01/01 · openalex publication_date 1997/01/01 · crossref created 2002/07/26 · openalex created_date 2016/06/24 · crossref deposited 2021/05/13 · crossref indexed 2026/05/12 · openalex updated_date 2026/07/23

Citations

• Rapid chromatographic technique for preparative separations with moderate resolution
• Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Cited by

• Ethisterone [wikipedia]