Nuclear receptor modulation – Role of coregulators in selective estrogen receptor modulator (SERM) actions

2014/06/16 by Qin Feng, Bert W. O’Malley · 65 citations
Biochemistry, Genetics and Molecular Biology · Chemistry · Medicine · #Agonist #Biochemistry #Breast cancer #Cancer #Cancer research #Chemistry #Cytokine Signaling Pathways and Interactions #Endocrinology #Estrogen #Estrogen and related hormone effects #Estrogen receptor #Estrogen receptor alpha #Estrogen-related receptor gamma #Inflammatory mediators and NSAID effects #Internal medicine #Medicine #Nuclear receptor #Pharmacology #Receptor #Selective estrogen receptor modulator #Tamoxifen #Transcription factor

paper · doi:10.1016/j.steroids.2014.06.008

published in Steroids 90, 39-43 (Elsevier BV)

openalex publication_date 2014/06/16 · crossref created 2014/06/16 · crossref issued 2014/11/01 · crossref published 2014/11/01 · crossref published-print 2014/11/01 · crossref deposited 2022/04/08 · openalex created_date 2025/10/10 · crossref indexed 2026/04/02 · openalex updated_date 2026/08/01

Citations

• Nuclear Receptor Coactivator ACTR Is a Novel Histone Acetyltransferase and Forms a Multimeric Activation Complex with P/CAF and CBP/p300
• Molecular Determinants for the Tissue Specificity of SERMs
• Activation of the Estrogen Receptor Through Phosphorylation by Mitogen-Activated Protein Kinase
• AIB1, a Steroid Receptor Coactivator Amplified in Breast and Ovarian Cancer
• Molecular basis of agonism and antagonism in the oestrogen receptor
• The Structural Basis of Estrogen Receptor/Coactivator Recognition and the Antagonism of This Interaction by Tamoxifen

Cited by

• Selective estrogen receptor modulator [wikipedia]