Structural Insights into the Mode of Action of a Pure Antiestrogen

2001/02/01 by A.C.W. Pike, Ashley C.W. Pike, A.Marek Brzozowski +9 · 9 citations
Biochemistry, Genetics and Molecular Biology · Medicine · Neuroscience · #Estrogen and related hormone effects #Menopause: Health Impacts and Treatments #Nuclear Receptors and Signaling

paper · pdf · doi:10.1016/s0969-2126(01)00568-8

crossref issued 2001/02/01 · crossref published 2001/02/01 · crossref published-print 2001/02/01 · openalex publication_date 2001/02/01 · crossref created 2002/07/25 · crossref deposited 2021/05/11 · openalex created_date 2025/10/10 · crossref indexed 2026/06/30 · openalex updated_date 2026/07/15

Citations

• PROCHECK: a program to check the stereochemical quality of protein structures

Cited by

• The 2.0 Å crystal structure of the ERα ligand‐binding domain complexed with lasofoxifene
• Selective estrogen receptor modulators (SERMs): Mechanisms of anticarcinogenesis and drug resistance
• Ser-884 Adjacent to the LXXLL Motif of Coactivator TRBP Defines Selectivity for ERs and TRs
• Coregulator Function: A Key to Understanding Tissue Specificity of Selective Receptor Modulators
• Antiestrogens and Selective Estrogen Receptor Modulators as Multifunctional Medicines. 2. Clinical Considerations and New Agents
• Reflections on the Discovery and Significance of Estrogen Receptor β
• Selective Estrogen-Receptor Modulators — Mechanisms of Action and Application to Clinical Practice
• Estrogen Receptors: Their Actions and Functional Roles in Health and Disease
• Antiestrogen [wikipedia]