The medicinal chemistry of carboranes

2002/10/01 by John F Valliant, John F. Valliant, Katharina J Guenther +8 · 30 citations
Chemistry · Medicine · #Bone health and treatments #Boron #Boron Compounds in Chemistry #Carborane #Chemistry #Combinatorial chemistry #Organic chemistry #Radiopharmaceutical Chemistry and Applications

paper · doi:10.1016/s0010-8545(02)00087-5

openalex publication_date 2002/10/01 · openalex created_date 2025/10/10 · openalex updated_date 2026/07/26

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• Synthesis of Polyhedral Borane Cluster Fused Heterocycles via Transition Metal Catalyzed B-H Activation. [europepmc]
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• Blue Emitting Star-Shaped and Octasilsesquioxane-Based Polyanions Bearing Boron Clusters. Photophysical and Thermal Properties. [europepmc]
• Carboranyl Derivatives of Rofecoxib with Cytostatic Activity against Human Melanoma and Colon Cancer Cells. [europepmc]
• Peptide-Drug Conjugates and Their Targets in Advanced Cancer Therapies. [europepmc]
• Addressing the Biochemical Foundations of a Glucose-Based "Trojan Horse"-Strategy to Boron Neutron Capture Therapy: From Chemical Synthesis to In Vitro Assessment. [europepmc]
• Synthesis and Structure of Nido -Carboranyl Azide and Its "Click" Reactions. [europepmc]
• Natural-Product-Directed Catalytic Stereoselective Synthesis of Functionalized Fused Borane Cluster-Oxazoles for the Discovery of Bactericidal Agents. [europepmc]
• Preparation of dendritic carboranyl glycoconjugates as potential anticancer therapeutics. [europepmc]
• Cobalt Bis-Dicarbollide Enhances Antibiotics Action towards Staphylococcus epidermidis Planktonic Growth Due to Cell Envelopes Disruption. [europepmc]
• Water-Stable Carborane-Based Eu 3+ /Tb 3+ Metal-Organic Frameworks for Tunable Time-Dependent Emission Color and Their Application in Anticounterfeiting Bar-Coding. [europepmc]
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• Synthesis and In Vitro Evaluation of a Set of 6-Deoxy-6-thio-carboranyl d-Glucoconjugates Shed Light on the Substrate Specificity of the GLUT1 Transporter. [europepmc]
• Carborane-Containing Hydroxamate MMP Ligands for the Treatment of Tumors Using Boron Neutron Capture Therapy (BNCT): Efficacy without Tumor Cell Entry. [europepmc]
• Sweet Battle of the Epimers─Continued Exploration of Monosaccharide-Derived Delivery Agents for Boron Neutron Capture Therapy. [europepmc]
• Towards the Application of Purely Inorganic Icosahedral Boron Clusters in Emerging Nanomedicine. [europepmc]
• In Vivo Application of Carboranes for Boron Neutron Capture Therapy (BNCT): Structure, Formulation and Analytical Methods for Detection. [europepmc]
• Nanostructured boron agents for boron neutron capture therapy: a review of recent patents. [europepmc]
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• Re-design and evaluation of diclofenac-based carborane-substituted prodrugs and their anti-cancer potential. [europepmc]
• Unraveling aromaticity: the dual worlds of pyrazole, pyrazoline, and 3D carborane. [europepmc]
• An Isolated Lithium ortho -Carboranyl Cuprate Complex for the Synthesis of Multiple-Carborane-Substituted Arenes from (Hetero)Aryl Bromides and Chlorides. [europepmc]